目的合成一种具有游离伯胺的卡莫司他衍生物。方法以对羟基苯乙酸为原料,经4步反应得到目标化合物。结果与结论成功制备了目标产物,所得产物的化学结构经^1HNMR、MS确认。
OBJECTIVE To synthesize a kind of Camostat derivatives with free primary amines. METHODS The target compound was synthesized via four steps with 4 - hydroxyphenylacetic acid. RESULTS and CONCLUSION The target compound was success- fully synthesized,and its chemical structure was conformed by ^1HNMR and MS.