中文摘要：

随着中药现代化研究的新进展，越来越多的研究表明许多中药中的化学成分只有经代谢后才具有生物活性．因此，对中药单体成分及复方的代谢化学研究引起了越来越多的研究人员的重视．近年来对代谢化学的研究逐步深入，中药代谢化学研究方法也随之深入，为中药化学成分及其产生生物活性的有效成分的研究提供依据．概述了有关代谢化学研究方法的新进展，为中药新药研究、中药药效物质研究、以中药有效成分为先导的药物研究及中药质量评价提供了依据．

英文摘要：

As the new progress of study on the modernization of traditional Chinese medicine, more and more researches show that its chemical composition only have biological activity af- ter metabolism. Therefore, research on metabolic chemistry of monomer components and com- pound prescription of Chinese medicine has caused more and more researchers＇ attention. Study on metabolic chemistry in recent years gradually thorough, and chemical research method of its metabolism with in - depth, then provides the basis for the research on its chemical composition and active ingredients of biological activity. This paper summarized the new progress of research method of metabolic chemistry, and provided a basis for the re- search on new drug, pharmaeodynamic material for traditional Chinese medicine, drug re- search on active ingredients of traditional Chinese medicinal for the pilot and quality evalua- tion of traditional Chinese medicine.