中文摘要：

吲哚二酮哌嗪类化合物是一类重要的杂环化合物,自然界中存在许多含有此结构单元的物质.由于该类物质具有多种生物活性,特别是抗肿瘤活性,因此它们的合成得到了广泛的研究.综述了吲哚二酮哌嗪类化合物的主要合成方法及其研究进展.

英文摘要：

Indolyl diketopiperazines are a very important class of heterocycles and widely found in the nature.Due to their broad range of bioactivities,especially anti-tumor activities,and their synthesis has attracted much attention.In this paper,the synthetic methods and their development are reviewed.