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Fluorescence Polarization for the Evaluation of Small-Molecule Inhibitors of PCAF-BRD/Tat-AcK50 Asso
ISSN号:1860-7179
期刊名称:ChemMedChem
时间:2014.6.8
页码:928-931
相关项目:化学小分子探针引导的细胞信号转导途径研究
作者:
汪志勇|
同期刊论文项目
化学小分子探针引导的细胞信号转导途径研究
期刊论文 66
同项目期刊论文
Small organic molecules targeting PCAF bromodomin as potent inhibitors of HIV-1 replication.
Biosynthesis of thiopeptide antibiotics and their pathway engineering.
Cytotoxic constituents from Cryptocarya maclurei.
Multiplexing of combinatiorial chemistry in antimycin biosynthesis: expansion of molecular diversity
Insight into bicyclic thiopeptide benifited from development of a uniform approach for molecular eng
Antitumor effect of naturally occurring oligomeric resveratrol derivatives.
Curvulamine, a Novel Antibacterial Alkaloid with New Extender Units from Curvularia sp. IFB-Z10. Wen
New flavonol and diterpenoids from the endophytic fungus Aspergillus sp. YXf3
Benzothiazoles exhibit broad-spectrum antitumor activity: their potency, structure-activity and stru
Insight into bicyclic thiopeptide benefited from development of a uniform approach for molecular eng
Discovery of a Negative Allosteric Modulator of GABAB Receptors. Lin-Hai Chen, Sun Bing, Yang Zhang,
Fumigaclavines D–H, New Ergot Alkaloids from Endophytic Aspergillus fumigatus. Jing Xu, Yong Chun So
Single-Cell Chemical Proteomics with an Activity-Based Probe: Identification of Low-Copy Membrane Pr
Cross-couplingtype tandem chloropalladation/dearomative cyclization towards functionalizedbridged [3
Modified Calanolides incorporated with furan-2-nitro mimics againstMycobacterium tuberculosis
Copper-catalyzed Ligand-free Amidation of Aryl iodides and Amino AcidAmides to Synthesize C3-(Z)-1H-
Copper/Silver-MediatedCascade Reactions for the Construction of 2-Sulfonylbenzo[b]furans from trans-
Iodine(III)-mediated[3+2] cyclization for one-pot synthesis of benzo[d]isoxazole-4,7-diol,benzodiiso
Catalyst-freesulfonylation of activated alkenes for highly efficient synthesis ofmono-substituted et
Goldnanoparticles supported on titanium dioxide: an efficient catalyst for highlyselective synthesis
Copper-CatalyzedEnantioselective Friedel-Crafts Alkylation of Pyrrole with Isatins
Agreen and efficient access to aryl nitriles via an electrochemical anodicoxidation
Copper-CatalyzedEnantioselective Hetero-Diels-Alder Reaction of Danishefsky?’s Diene withβ,γ-Unsatur
Copper CatalyzedEnantioselective Alkylation of Pyrrole with β,γ-Unsaturated α-Ketoesters:Application
Supportedgold-catalyzed and ammonia-promoted selective synthesis of quinazolines inaqueous media
Cerium(III)-catalyzedcascade cyclization: an efficient approach to functionalizedpyrrolo[1,2-a]quino
Cyclization of polyketidesand non-ribosomal peptides on and off their assembly lines,
Aromatic PolyketidesProduced by Bacterial Iterative Type I Polyketide Synthases
Pictet–Spengler reaction based biosyntheticmachinery in fungi
Highly Enantioselective Construction of Fluoroalkylated QuaternaryStereocenters viaOrganocatalytic D
Bismuth nanoparticles: an efficient catalyst for reductive coupling of nitroarenes toazo-compounds
Cyclization of polyketidesand non-ribosomal peptides on and off their assembly linesEffect of Stereo
Efficient synthesis of 2-arylquinazolines via copper-catalyzed dual oxidative benzylicC-H aminations
Highly Diastereo- and Enantioselective Michael Addition of Nitroalkanes to2-Enoyl-Pyridine N-Oxides
Copper-CatalyzedRadical Methylation/C-H Amination/Oxidation Cascade for the Synthesis ofQuinazolinon
Electrosynthesis of enaminones directly from methylketones and amines with nitromethane as a carbon
以生物合成为基础的红霉素A的产量提高和结构改造
Regio-controlled synthesis of unsymmetrical pyrazine-fused sinomenine derivatives and discriminate s
An enzymatic [4+2]cyclization cascade creates the pentacyclic core of pyrroindomycins
Thiopeptide AntibioticsExhibit a DualModeof Action against Intracellular Pathogens by Affecting Both
Direct Electrosynthesis of Ketones from BenzylicMethylenes by Electrooxidative CH Activation
Targeting the γ-/β-secretase interaction reducesβ-amyloid generation and ameliorates Alzheimer’s dis
基于活性小分子探针的蛋白质标记基于活性小分子探针的蛋白质标记 (第9章),化学生物学前沿与展望(蒋华良等编)
Synthesisof benzofused five-ring sultams via Rh-catalyzed CH olefination directed by anN-Ac substitu
Metabolic coupling of twosmall-molecule thiols programs the biosynthesis of lincomycin A
A simple and efficient approach to realize difunctionalization of arylketoneswith malonate esters vi
Oxidative coupling of methylamine with an aminylradical: direct amidation catalyzed by I2/TBHP with
An efficient synthesis of amides from alcohols andazides catalyzed by a bifunctional catalyst Au/DNA
Electrochemical Synthesis of the Arylα-Ketoesters fromAcetophenones Mediated by KI
Cobalt-catalyzed oxidative[3+2] cycloadditionreactions: an efficient synthesis of pyrrolo- and imida
A novel approach for the one-pot preparation ofα-ketoamides by anodic oxidation
Metal-Organic Framework with Functional Amide Groupsfor Highly Selective Gas Separation
Discovery and efficientsynthesis of a biological active alkaloid inspired by thiostrepton biosynthes
Spiroketal formation andmodification in avermectin biosynthesis involves a dual activity of AveC
FK506 maturation involves acytochrome P450 protein-catalyzed four electron oxidation in parallel wit
Bifunctional Amino Sulfonohydrazide Catalyzed Direct Asymmetric MannichReaction of Cyclic Ketimines
CuI-catalyzed and air promoted oxidativecyclization for one-pot synthesis of polyarylated oxazoles
Synthesis of Chromones through LiOtBu/Air-Mediated Oxidation and Regioselective Cyclization ofo-Hydr
便捷、高效、可实现放大合成mycothiol的全合成策略研究
适用于荧光成像的化学发色团与生物正交反应研究进展
大环内酯类免疫抑制剂他克莫司的生物合成机制研究进展
Synthetic Analogues of Betulinic Acid as Potent Inhibitors of PS1/BACE1 Interaction to Reduce Aβ Generation