几新奇的 N-[(1-ferrocenylethylidene ) 氨基]-N -- D-glycopyranosylthioureas 高效地经由一个六步的过程被综合了,作为分别地开始材料利用三 monosaccharides (D 葡萄糖, D 半乳糖和 D 木糖) 。他们 preliminarily 决心对某些真菌显示生物活动。目标混合物被分光镜的方法和元素的分析明白地描绘了。一条开始其他的合成线路,看起来合理,由于它的无效被排除了。
Several novel N′-[(1-ferrocenylethylidene)amino]-N′-β-D-glycopyranosylthioureas have been efficiently synthesized via a six-step procedure, utilizing three monosaccharides (D-glucose, D-galactose and D-xylose) as starting materials, respectively. They have been preliminarily determined to display biological activity against certain fungi. The target compounds have been unambiguously characterized by spectroscopic method and elemental analysis. An initially alternative synthetic route, which was seemingly reasonable, has been excluded due to its inefficiency.