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Palladium-Catalyzed Intramolecular Aminofluorination of Styrenes
  • ISSN号：1001-604X
  • 期刊名称：《中国化学：英文版》
  • 时间：0
  • 分类：TQ463.4[化学工程—制药化工] TP381[自动化与计算机技术—计算机系统结构;自动化与计算机技术—计算机科学与技术]
  • 作者机构：[1]State Key Laboratory of Organometallics Chemistry and Shanghai Mass Spectrometry Center, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, 354 Fenglin Road, Shanghai 200032, China
  • 相关基金：Project supported by the National Basic Research Program of China （No. 973-2011CB808700）, the National Natural Science Foundation of China （Nos. 20821002, 20872155, 20972175 and 20923005） and the ＂Hundred Talent Project＂ of the Chinese Academy of Sciences.
作者： 徐涛[1], 邱水发[1], 刘国生[1]
关键词： 氧化苯乙烯, 分子内, 钯催化, 氟化剂, 衍生物, 反应, palladium, intramoleclular, aminofluorination, fluoropyrrolidine
中文摘要：

新奇催化钯的 intramolecular 苯乙烯的氧化 aminofluorination 被把 NFSI 用作氟化开发了试剂。这反应为 2-aryl-3-fluoropyrrolidine 衍生物的合成代表了一个有效方法。

英文摘要：

A novel palladium-catalyzed intramolecular oxidative aminofluorination of styrenes has been developed by using NFSI as fluorinating reagent. This reaction represented an efficient method for the synthesis of 2-aryl-3-fluoropyrrolidine derivatives.

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期刊信息
  • 《中国化学：英文版》
  • 主管单位:
  • 主办单位:中国化学会
  • 主编：
  • 地址：上海市枫林路354号中科院上海有机化学研究所
  • 邮编：200032
  • 邮箱：
  • 电话：021-54925243
  • 国际标准刊号：ISSN：1001-604X
  • 国内统一刊号：ISSN：31-1547/O6
  • 邮发代号:4-646
  • 获奖情况:
  • 中国期刊方阵“双高”期刊
  • 国内外数据库收录:
  • 美国化学文摘（网络版）,荷兰文摘与引文数据库,美国科学引文索引（扩展库）,日本日本科学技术振兴机构数据库,英国英国皇家化学学会文摘
  • 被引量:175