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Synthesis of Potential Inhibitiors for Stat-3 Dimerization
  • ISSN号：1001-604X
  • 期刊名称：《中国化学：英文版》
  • 时间：0
  • 分类：R979.1[医药卫生—药品;医药卫生—药学]
  • 作者机构：[1]State Key Laboratory of Bio-organic and Natural Products Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai 200032, China, [2]Department of Chemistry, Northwest University, Xi'an, Shaanxi 710069, China, [3]Departments of Internal Medicine and Medicinal Chemistry, University of Michigan, Ann Arbor, M148109, USA
  • 相关基金：Project supported by the National Natural Science Foundation of China （Nos of Sciences （No. KGCX2-SW-209）. Dedicated to Professor Xikui Jiang on the occasion of his 80th birthday 20025207, 20272071, 20372075, 20321202） and the Chinese Academy
作者： 崔家荣[1], 简亚军[1,2], 伍贻康[1], 王少萌[3]
关键词： 抑制剂, 抗癌制剂, 苯炔, 芳香族, inhibitor, antitumor agent, benzyne, aromatics, angucyclinone
中文摘要：

九 bioactive ochromycinone 类似物通过线路的二种不同类型被综合。一些意外产品在导致相片的氧化被获得。此处揭示的综合体在文学补充那些并且包含其大多数以前在完全不同的上下文是学习的年的已知的中介把便宜存取提供给许多。

英文摘要：

Nine bioactive ochromycinone analogues were synthesized through two different types of routes. Some unexpected products were obtained in the photo-induced oxidation. The syntheses disclosed herein complement those in the literature and offer inexpensive access to many of the known intermediates involved, most of which were studied years ago in completely different contexts.

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期刊信息
  • 《中国化学：英文版》
  • 主管单位:
  • 主办单位:中国化学会
  • 主编：
  • 地址：上海市枫林路354号中科院上海有机化学研究所
  • 邮编：200032
  • 邮箱：
  • 电话：021-54925243
  • 国际标准刊号：ISSN：1001-604X
  • 国内统一刊号：ISSN：31-1547/O6
  • 邮发代号:4-646
  • 获奖情况:
  • 中国期刊方阵“双高”期刊
  • 国内外数据库收录:
  • 美国化学文摘（网络版）,荷兰文摘与引文数据库,美国科学引文索引（扩展库）,日本日本科学技术振兴机构数据库,英国英国皇家化学学会文摘
  • 被引量:175